CP 47,497

CP 47,497
Pravni status
Pravni status
  • Ilegalan u Nemačkoj i Francuskoj, Klasa B (UK)
Identifikatori
CAS broj70434-82-1 Зелена квачицаДа
70434-92-3 (C8 homolog)
ATC kodnone
PubChemCID 125835
ChEMBLCHEMBL163701 Зелена квачицаДа

CP 47,497 ili (C7)-CP 47,497 je agonist kanabinoidnog receptora, koji je razvilo preduzeće Pfizer tokom 1980-tih.[1] Ovaj materijal ima analgetsko dejstvo i koristi se u naučnim istraživanjima. Ono je potentan CB1 agonist sa Kd vrednošću od 2,1 nM.[2][3][4]

Vidi još

Reference

  1. ^ Weissman, A.; Milne, G. M.; Melvin Jr, L. S. (1982). „Cannabimimetic activity from CP-47,497, a derivative of 3-phenylcyclohexanol”. The Journal of Pharmacology and Experimental Therapeutics. 223 (2): 516—523. PMID 6290642. doi:10.1016/S0022-3565(25)33364-1. 
  2. ^ Shim, J. Y.; Welsh, W. J.; Howlett, A. C. (2003). „Homology model of the CB1 cannabinoid receptor: Sites critical for nonclassical cannabinoid agonist interaction”. Biopolymers. 71 (2): 169—189. PMID 12767117. doi:10.1002/bip.10424. 
  3. ^ Roger Pertwee. Cannabinoids. Handbook of Experimental Pharmacology Volume 168. Springer. ISBN 978-3-540-22565-2.
  4. ^ Little PJ, et al. „Pharmacology and stereoselectivity of structurally novel cannabinoids in mice”. Journal of Pharmacology and Experimental Therapeutics. 247: 1046—1051. 1988. .

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